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FR 139317
SynDRA canonical compound SYN1994330 — structure-anchored drug synonym record
| Primary target(s) | EDNRA |
|---|
| Mechanism of action | Endothelin receptor antagonist |
|---|
All known targets
Mechanisms of action (all sources)
- Endothelin receptor antagonist
- EDNRA INVERSE AGONIST
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ADGRF1
- GPR119
- HDAC6
- HRH1
- HRH2
- HSD17B10
- HTR1B
- HTR2A
- HTR2B
- HTR3A
- MBD4
- MPG
- MUTYH
- NEIL1
- NEIL2
- OGG1
- OPRK1
- OPRM1
- S1PR1
- SIGMAR1
- SLC17A5
- SLC6A3
- TDG
- TMEM97
- TSPO
- GPR35
- GLP1R
- ADRA1A
- FPR2
- ADRA1B
- ADRA2A
- ADRA2C
- ADRB1
- ADRB2
- ADRB3
- AGTR1
- APLNR
- C5AR1
- CHRM1
- CHRM4
Cross-references
Synonyms
- FR139317
- RefChem:141430
- C33H44N6O5
- PD 147953
- Tocris-1210
- GTPL998
- orb1704524
- SCHEMBL2124350
- HMS3412O03
- HMS3676O03
- SFA37560
- BDBM50286804
- MFCD00467722
- AKOS024456467
- NCGC00025042-01
- NCGC00025042-02
- AS-85708
- HY-102092
- G78199
- T22791
- SR-01000597371
- SR-01000597371-1
- BRD-K19318328-001-01-3
- FR-139317
- CHEBI:91886
- HMS3267B17
- BRD-A80641450-001-01-4
- 2-[[2-[[2-[[1-azepanyl(oxo)methyl]amino]-4-methyl-1-oxopentyl]amino]-3-(1-methyl-3-indolyl)-1-oxopropyl]amino]-3-(2-pyridinyl)propanoic acid
- L000260
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