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mubritinib
SynDRA canonical compound SYN0048265 — structure-anchored drug synonym record
| Primary target(s) | ERBB2 |
| Mechanism of action | Receptor tyrosine protein kinase inhibitor |
All known targets
Mechanisms of action (all sources)
- Receptor tyrosine protein kinase inhibitor
- ERBB2 INHIBITOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ADGRF1
- GRM6
- TDG
- SMUG1
- S1PR1
- OGG1
- NTHL1
- NEIL2
- NEIL1
- MUTYH
- MBD4
- KCNH2
- HDAC6
- GRM8
- GRM7
- GRM4
- ADRA2A
- GRM3
- GRM2
- GRM1
- GPR35
- GPR119
- GLP1R
- FPR2
- FFAR4
- CX3CR1
- C5AR1
- APLNR
- AGTR1
- ADRB2
- UNG
Cross-references
Synonyms
- C25H23F3N4O2
- ZTFBIUXIQYRUNT-UHFFFAOYSA-N
- SCHEMBL571874
- HMS3655P10
- HMS3744I11
- SB19375
- NCGC00346582-01
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