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cetrorelix
SynDRA canonical compound SYN0041819 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | GNRH1 | GNRHR | LHCGR |
|---|
| Mechanism of action | gonadotropin releasing factor hormone receptor antagonist |
|---|
| Indication | premature luteinizing hormone surges |
|---|
| Disease area | endocrinology |
|---|
All known targets
Mechanisms of action (all sources)
- GNRHR ANTAGONIST
- Gonadotropin-releasing hormone receptor antagonist
- gonadotropin releasing factor hormone receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ABCB11
- MRGPRX2
- HTR1A
- SLC6A4
- SLC6A3
- SLC6A2
- PTGS1
- PGR
- PDE4A
- PDE3A
- OPRM1
- MAOA
- HTR2B
- HRH3
- ACHE
- HDAC6
- F2
- ESR1
- DRD3
- DRD1
- CHRM2
- CHRM1
- AR
- ADRA2A
- ADRA1A
- ADORA1
- TBXA2R
Drug classes
- Gonadotropin Releasing Hormone Receptor Antagonists
- Fertility Agents, Female
- Hormone Antagonists
- Reproductive Control Agents
- Gonadotropin Releasing Hormone Receptor Antagonist
ATC classes
- H01C · HYPOTHALAMIC HORMONES
Cross-references
Synonyms
- CETRORELIX ACETATE
- CETROTIDE
- Cetrotide
- cetrotide
- cetrorelix acetate
- Cetrorelixum
- Cetrorelix (INN)
- Cetrotide (TN)
- HS-2008
- Ac-D-Nal(2)-D-Phe(pCl)-D-Pal(3)-Ser-Tyr-D-Cit-Leu-Arg-Pro-D-Ala-NH2
- OON1HFZ4BA
- SB 75
- CHEBI:59224
- RefChem:58062
- DTXCID5020996
- H01CC02
- Cetrorelixum [INN-Latin]
- Cetrorelix [INN]
- C70H92ClN17O14
- Cetrelix Acetate
- SB-075
- Cetrorelix [INN:BAN]
- UNII-OON1HFZ4BA
- HSDB 7696
- Antide acetate salt
- CETRORELIX [MI]
- CETRORELIX [HSDB]
- CETRORELIX [VANDF]
- CETRORELIX [WHO-DD]
- SCHEMBL61331
- CETRORELIX [EMA EPAR]
- GTPL1190
- CETRORELIX [ORANGE BOOK]
- SCHEMBL19712202
- SCHEMBL19712205
- SCHEMBL29397892
- SCHEMBL29406896
- SCHEMBL29887354
Reported adverse events
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