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VALETHAMATE
SynDRA canonical compound SYN0033752 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | CHRM1 | CHRM4 | CHRM5 |
|---|
| Mechanism of action | acetylcholine receptor antagonist |
|---|
| Indication | labor induction |
|---|
| Disease area | obstetrics/gynecology |
|---|
All known targets
- CHRM1
- CHRM4
- CHRM5
- CHRM2
- CHRM3
- CYP2D6
- SIGMAR1
Mechanisms of action (all sources)
- acetylcholine receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ACHE
- LCK
- MMP1
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- MAPK1
- MAOA
- KCNH2
- ADORA1
- HTR6
- HTR2C
- HTR2B
- HTR2A
- HRH2
- HRH1
- HMGCR
- HDAC6
- MMP9
- NPY1R
- NPY2R
- NR3C1
- TDP1
- TBXAS1
- TACR2
- TACR1
- SLC6A4
- SLC6A3
- SLC6A2
- PTPRC
- PTGS2
- PTGS1
- PTAFR
- PRKCA
- PPP3CA
- PDE5A
- OPRM1
- OPRK1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
ATC classes
- A03A · DRUGS FOR FUNCTIONAL GASTROINTESTINAL DISORDERS
Cross-references
Synonyms
- valethamate bromide
- Valethamate cation
- Valethamate ion
- D64S64QVX7
- RefChem:193564
- UNII-D64S64QVX7
- Murel
- Epidosan
- NCGC00185757-01
- Letamate
- Velamate
- Elist
- Release V
- VALETHAMATE [WHO-DD]
- SCHEMBL249537
- CHEBI:135303
- UPPMZCXMQRVMME-UHFFFAOYSA-N
- FH171076
- NS00008564
- BRD-A56613951-004-01-1
- Resitan
- AC-19311
- DB-057189
- F242202
- Valethamate Bromide
- Shinmetane (TN)
- DTXCID0028953
- Valethamate bromide
- Epidosin
- Epidozin
- AKOS015902836
- SR-01000883681-1
- HMS5084C15
- Valethamatbromid
- VALETHAMATE BROMIDE [MI]
- EBC-157238
- GLXC-08172
- VALETHAMATE BROMIDE [WHO-DD]
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