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AZASETRON
SynDRA canonical compound SYN0025633 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | HTR3A |
|---|
| Mechanism of action | Serotonin receptor antagonist |
|---|
| Indication | genitial herpes |
|---|
| Disease area | infectious disease |
|---|
All known targets
Mechanisms of action (all sources)
- Serotonin receptor antagonist
- HTR3A ANTAGONIST
- HTR3B ANTAGONIST
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- KCNH2
- PDE4D
- ACHE
- MMP1
- MLNR
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- MAPK1
- MAOA
- LCK
- KAT2A
- NPY1R
- HTR6
- HTR2C
- HTR2B
- HTR2A
- HTR1A
- HRH3
- HRH2
- HRH1
- HMGCR
- HDAC6
- GHSR
- MMP9
- NPY2R
- ADORA1
- NR1I2
- TDP1
- TBXAS1
- TBXA2R
- TACR2
- TACR1
- SLC6A4
- SLC6A3
- SLC6A2
- SLC29A1
- SIGMAR1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Antiemetics
- Central Nervous System Agents
- Gastrointestinal Agents
- Neurotransmitter Agents
- Peripheral Nervous System Agents
- Serotonin Agents
- Serotonin Antagonists
Cross-references
Synonyms
- azasetron hydrochloride
- nazasetron
- azasetron HCl
- Y-25130
- Nazasetron
- Azasetron [INN]
- C17H20ClN3O3
- WUKZPHOXUVCQOR-UHFFFAOYSA-N
- Azasetron (INN)
- 6-Chloro-4-methyl-3-oxo-N-(quinuclidin-3-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carboxamide
- NCGC00024563-02
- DSSTox_RID_81029
- DSSTox_CID_25651
- DSSTox_GSID_45651
- (- )-6-Chloro-3,4-dihydro-4-methyl-3-oxo-N-3-quinuclidinyl-2H-1,4-benzoxazine-8-carboxamide
- N-(1-azabicyclo[2.2.2]octan-3-yl)-6-chloro-4-methyl-3-oxo-1,4-benzoxazine-8-carboxamide
- WR85915
- Azasetron HCl
- Serotone
- Azasetron (hydrochloride)
- Y-25130 hydrochloride
- C17H20ClN3O3.HCl
- Azasetron hydrochloride [JAN]
- 6-chloro-4-methyl-3-oxo-N-(quinuclidin-3-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carboxamide hydrochloride
- Azasetron hydrochloride (JAN)
- N-(1-azabicyclo[2.2.2]octan-3-yl)-6-chloro-4-methyl-3-oxo-1,4-benzoxazine-8-carboxamide hydrochloride
- 2H-1,4-Benzoxazine-8-carboxamide, 3,4-dihydro-N-1-azabicyclo(2.2.2)oct-3-yl-6-chloro-
- DTXCID5025651
- azasetronum
- RefChem:115971
- (R)-Azasetron
- Y 25130
- CAS-123040-69-7
- seroton
- AZASETRON [MI]
- Biomol-NT_000105
- UNII-77HC7URR9Z
- AZASETRON [WHO-DD]
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