← SynDRA

PICOTAMIDE

SynDRA canonical compound SYN0024733 — structure-anchored drug synonym record

All known targets

• TBXA2R
• TBXAS1

Mechanisms of action (all sources)

• Thromboxane synthase inhibitor
• Thromboxane receptor antagonist
• TBXAS1 INHIBITOR
• Thromboxane-A synthase inhibitor
• TBXA2R INHIBITOR
• Thromboxane A2 receptor inhibitor

Bioactivity evidence (ChEMBL activities table — not curator-asserted)

• ADORA1
• MLNR
• HDAC6
• HRH1
• HRH2
• HRH3
• HTR1A
• HTR2A
• HTR2B
• HTR2C
• HTR3A
• KCNH2
• L3MBTL1
• MAOA
• MC3R
• NPY1R
• EDNRA
• NR1I2
• NR3C1
• OPRD1
• OPRK1
• OPRM1
• PDE3A
• PDE4D
• PGR
• PIN1
• PTGS2
• SLC6A3
• SLC6A4
• SMAD3
• GHSR
• DRD3
• ADORA2A
• BLM
• ADORA3
• ADRA1A
• ADRA2A
• ADRA2B
• ADRA2C
• ADRB1

Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)

• CP1A2
• CP3A4
• ITA4

Drug classes

• Hematologic Agents
• Platelet Aggregation Inhibitors

ATC classes

• B01A · ANTITHROMBOTIC AGENTS

Cross-references

• PubChem CID: 4814
• ChEMBL: CHEMBL1257015
• DrugBank: DB13327
• ChEBI: CHEBI:93175
• KEGG: D07140
• Wikipedia: Picotamide
• LINCS BRD: BRD-K67277431

Synonyms

• picotamide monohydrate
• picotamide hydrate
• G-137
• NSC-304384
• G 137
• NSC 304384
• RefChem:174171
• DTXCID50108989
• 4-methoxy-N1,N3-bis(pyridin-3-ylmethyl)isophthalamide
• EINECS 251-245-7
• Picotamide [INN:BAN]
• BRN 0499268
• UNII-654G2VCI4Q
• SR-01000076086
• N,N'-Bis(3-picolyl)-4-methoxyisophthalamide
• 4-Methoxy-N,N'-bis(3-pyridylmethyl)isophthalamide
• Picotamide (BAN)
• 4-Methoxy-N,N'-bis(3-pyridylmethyl)isophthaldiamide
• Isophthalamide, 4-methoxy-N,N'-bis(3-pyridylmethyl)-
• PICOTAMIDE [MI]
• Prestwick0_000119
• Prestwick1_000119
• Prestwick2_000119
• Prestwick3_000119
• Lopac-P-8477
• PICOTAMIDE [MART.]
• PICOTAMIDE [WHO-DD]
• Lopac0_001003
• BSPBio_000138
• N,N'-Bis(3-pyridylmethyl)-4-methoxyisophthalamide
• SCHEMBL137025
• SPBio_002077
• BPBio1_000152
• orb1298325
• SCHEMBL30206880
• SCHEMBL30254057
• CHEBI:93175
• GTPL11379