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TOCAINIDE
SynDRA canonical compound SYN0020321 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · OTC |
|---|
| Primary target(s) | SCN5A |
|---|
| Mechanism of action | Sodium channel blocker |
|---|
| Indication | cardiac arrythmia |
|---|
| Disease area | cardiology |
|---|
All known targets
- SCN5A
- SCN10A
- SCN11A
- SCN1A
- SCN2A
- SCN3A
- SCN4A
- SCN7A
- SCN8A
- SCN9A
Mechanisms of action (all sources)
- Sodium channel blocker
- SCN1A BLOCKER
- Sodium channel alpha subunit blocker
- SCN5A BLOCKER
- SCN4A BLOCKER
- SCN7A BLOCKER
- SCN2A BLOCKER
- SCN9A BLOCKER
- SCN3A BLOCKER
- SCN11A BLOCKER
- SCN8A BLOCKER
- SCN10A BLOCKER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ACHE
- HTR5A
- MLNR
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- MAPK1
- MAOA
- LCK
- KCNH2
- HTR7
- HTR6
- HTR3A
- MMP9
- HTR2C
- HTR2B
- HTR2A
- HTR1A
- HRH3
- HRH2
- HRH1
- HMGCR
- HDAC6
- GIPR
- GHSR
- GCGR
- MMP1
- NPY1R
- FYN
- PTGS1
- TBXAS1
- TBXA2R
- TACR2
- TACR1
- SLC6A4
- SLC6A3
- SLC6A2
- SLC29A1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- 5HT2A
- KCMB2
- RAPGEF3
- RPGF3
Drug classes
- Anti-Arrhythmia Agents
- Cardiovascular Agents
- Membrane Transport Modulators
- Sodium Channel Blockers
- Voltage-Gated Sodium Channel Blockers
ATC classes
- C01B · ANTIARRHYTHMICS, CLASS I AND III
Cross-references
Synonyms
- TONOCARD
- tocainide hydrochloride
- (RS)-Tocainide
- (+/-)-Tocainide
- DL-Tocainide
- tocainide HCl
- Tocainida
- W-36095
- Taquidil
- Tocainidum
- Tonocard
- Astra W 36095
- Tocainida [INN-Spanish]
- Tocainidum [INN-Latin]
- Tocainide (USAN/INN)
- Tocainide [USAN:BAN:INN]
- Alanyl-2,6-xylidide
- 2-Amino-2',6'-propionoxylidide
- W 36095
- CHEBI:9611
- RefChem:898536
- DTXCID7020766
- C01BB03
- W36095
- MFCD00072010
- 2',6'-Propionoxylidide, 2-amino-
- SMR000466388
- EINECS 255-505-0
- UNII-27DXO59SAN
- BRN 2416564
- Tocainide [USAN:INN:BAN]
- Tocainide?
- TOCAINIDE [INN]
- TOCAINIDE [MI]
- TOCAINIDE [USAN]
- Prestwick0_001027
- Prestwick1_001027
- Prestwick2_001027
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