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DESOGESTREL
SynDRA canonical compound SYN0008940 — structure-anchored drug synonym record
| Clinical phase | Launched |
| Approval status | Approved · Rx/OTC |
| Primary target(s) | ESR1 | PGR |
| Mechanism of action | progesterone receptor agonist |
| Indication | contraceptive |
| Disease area | endocrinology |
All known targets
Mechanisms of action (all sources)
- PGR AGONIST
- PGR MODULATOR
- PGR BINDER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- NR3C1
- NR1I2
- ADORA3
- SLC6A4
- SLC6A2
- CHRM2
- DRD3
- AR
- MAOA
- NPY1R
- MLNR
- MC3R
- ACHE
- HTR3A
- HTR2C
- HTR2B
- HTR2A
- KCNH2
- OPRK1
- OPRD1
- HRH3
- OPRM1
- PDE3A
- PDE4A
- PDE4D
- PTGS1
- PTGS2
- SLC29A1
- SLC6A3
- TBXA2R
- HTR1A
- HDAC6
- HRH2
- CCKAR
- ADORA2A
- ADRA1A
- ADRA2A
- ADRA2B
- ADRA2C
- ADRB1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Progestin
- Contraceptive Agents
- Contraceptive Agents, Female
- Contraceptive Agents, Hormonal
- Contraceptives, Oral, Hormonal
- Contraceptives, Oral, Synthetic
- Hormones
- Progestins
- Reproductive Control Agents
ATC classes
- G03A · HORMONAL CONTRACEPTIVES FOR SYSTEMIC USE
- PROGESTOGENS AND ESTROGENS IN COMBINATION
Cross-references
Synonyms
- AVERI
- BEKYREE
- CYCLESSA
- DESOGEN
- DESOGESTREL AND ETHINYL ESTRADIOL
- EMOQUETTE
- ENSKYCE
- ISIBLOOM
- KALLIGA
- KARIVA
- KIMIDESS
- MIRCETTE
- Org 2969
- cerazette
- Mircette
- ORG-2969
- Aizea
- Cerazette
- Cerelle
- Desogestrel component of bekyree
- Desogestrel component of cyclessa
- Desogestrel component of desogen
- Desogestrel component of enskyce
- Desogestrel component of isibloom
- Desogestrel component of kariva
- Desogestrel component of mircette
- Desogestrel component of ortho-cept
- Desogestrel component of pimtrea
- Desogestrel component of velivet
- Desogestrel component of viorele
- Desogestrel component of volnea
- Desomono
- Feanolla
- Nacrez
- Zelleta
- Desogen
- Desogestrelum
- Organon Brand of Desogestrel
Reported adverse events
- Migraine
- Nausea
- Vomiting
- Thrombophlebitis
- Erythema multiforme
- Erythema nodosum
- Hirsutism
- Nervousness
- Rash
- Cerebral thrombosis
- Myocardial infarction
- Headache
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