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TELENZEPINE
SynDRA canonical compound SYN0008473 — structure-anchored drug synonym record
| Clinical phase | Phase 3 |
|---|
| Primary target(s) | CHRM1 |
|---|
| Mechanism of action | Acetylcholine receptor antagonist |
|---|
All known targets
Mechanisms of action (all sources)
- Acetylcholine receptor antagonist
- CHRM1 MODULATOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ALDH1A1
- APEX1
- SLCO1B3
- SLCO1B1
- SAMHD1
- LMNA
- L3MBTL1
- GALC
- EHMT2
- DRD1
- CYP3A4
- CYP2D6
- CYP2C9
- CYP2C19
- CYP1A2
- CBX1
- BAZ2B
- TSHR
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ACM1
- ACM4
- ACM5
- CP2C9
- CP2CJ
- CP2D6
- CP3A4
- KCNJ1
- MDR1
Drug classes
Cross-references
Synonyms
- Telenzepina
- NSC-758679
- Telenzepine [INN]
- Telenzepinum [Latin]
- Telenzepino [Spanish]
- UNII-0990EG3K10
- 0990EG3K10
- NCGC00015987-05
- DSSTox_RID_80752
- DSSTox_CID_25209
- 1-methyl-10-[2-(4-methylpiperazin-1-yl)acetyl]-5H-thieno[3,4-b][1,5]benzodiazepin-4-one
- DSSTox_GSID_45209
- 4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-10H-thieno(3,4-b)(1,5)benzodiazepin-10-one
- Telenzepine hydrochloride
- Telenzepine dihydrochloide
- C19H22N4O2S
- Telenzepino
- Telenzepinum
- Telenzepine dihydrochloride hydrate
- BY-802
- [3H](+)telenzepine
- NSC 758679
- DTXCID3025209
- RefChem:932670
- TELENZEPINE 2HCL
- (+/-)-Telenzepine
- CAS-80880-90-6
- ()-Telenzepine
- VSWPGAIWKHPTKX-UHFFFAOYSA-N
- Tocris-1122
- Lopac-T-122
- TELENZEPINE [MI]
- Prestwick0_000303
- Prestwick1_000303
- Prestwick2_000303
- Prestwick3_000303
- Spectrum3_001839
- TELENZEPINE [MART.]
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