← SynDRA
FLUPIRTINE
SynDRA canonical compound SYN0007919 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | KCNQ2 |
|---|
| Mechanism of action | Glutamate receptor antagonist |
|---|
| Indication | pain relief |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- KCNQ2
- KCNQ1
- KCNQ3
- ADRA2A
- SHMT2
Mechanisms of action (all sources)
- Glutamate receptor antagonist
- KCNQ2 MODULATOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- KCNH2
- KCNQ4
- ESR1
- PTGS2
- ABCB11
- MAPT
- NR3C1
- NR1I2
- NPY1R
- NFKB1
- NFE2L2
- MPHOSPH8
- MLNR
- MC3R
- MBNL1
- MAOA
- MAPK1
- OPRK1
- L3MBTL1
- KMT2A
- KDM4E
- KDM4A
- IDH1
- HTR3A
- HTR2C
- HTR2B
- HTR2A
- OPRD1
- OPRM1
- HSD17B10
- PDE3A
- USP2
- USP1
- TSG101
- TDP1
- TBXA2R
- TARDBP
- SMPD1
- SMAD3
- SLC6A4
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ADCY9
- ALAT2
- SYK
- RPGF4
- PNMT
- NTM1A
- NNMT
- KSYK
- KCNQ5
- HNMT
- GNMT
- GLSK
- GAMT
- FUMH
- ESRRA
- CP3A7
- CP3A4
- CP2D6
- CP2CJ
- CP2C9
- COMT
- TP53
Drug classes
- Analgesics
- Central Nervous System Agents
- Peripheral Nervous System Agents
- Sensory System Agents
ATC classes
- N02B · OTHER ANALGESICS AND ANTIPYRETICS
Cross-references
Synonyms
- flupirtin maleate
- flupirtine maleate
- katadolon
- Flupirtina
- Flupirtinte
- W-2964
- Flupirtine [INN:BAN]
- Flupirtinum [INN-Latin]
- Flupirtino [INN-Spanish]
- UNII-MOH3ET196H
- C15H17FN4O2
- EINECS 260-503-8
- MOH3ET196H
- JUUFBMODXQKSTD-UHFFFAOYSA-N
- ethyl N-[2-amino-6-[(4-fluorophenyl)methylamino]pyridin-3-yl]carbamate
- D 9998
- ethyl 2-amino-6-(4-fluorobenzylamino)pyridin-3-ylcarbamate
- Flupirtinum
- Flupirtino
- MLS002153180
- Carbamic acid, (2-amino-6-(((4-fluorophenyl)methyl)amino)-3-pyridinyl)-, ethyl ester
- NCGC00015451-03
- SMR001230672
- Flupirtin
- Carbamic acid, [2-ami
- flupirtina
- ethyl 2-amino-6-((p-fluorobenzyl)amino)-3-pyridinecarbamate
- RefChem:141020
- DTXCID4028410
- N02BG07
- Flupirtine (INN)
- FLUPIRTINE [INN]
- NCGC00015451-01
- FLUPIRTINE [MI]
- Lopac-F-8927
- FLUPIRTINE [VANDF]
- FLUPIRTINTE [VANDF]
- FLUPIRTINE [WHO-DD]
Look up FLUPIRTINE in the interactive SynDRA portal →