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MEPAZINE
SynDRA canonical compound SYN0007583 — structure-anchored drug synonym record
| Clinical phase | Phase 2 |
|---|
| Primary target(s) | MALT1 |
|---|
| Mechanism of action | MALT1 inhibitor |
|---|
All known targets
- MALT1
- ADRA1D
- GFER
- SIGMAR1
- Pgrmc1
- HTR6
- HTR2C
- HTR2B
- HTR2A
- HRH1
- DRD3
- ADRA2A
Mechanisms of action (all sources)
- MALT1 INHIBITOR
- Mucosa-associated lymphoid tissue lymphoma translocation protein 1 inhibitor
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- DRD1
- OPRM1
- ESR1
- KCNH2
- ABCB11
- NPY1R
- MMP9
- MMP1
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK1
- MAPK14
- NR3C1
- MAOA
- LCK
- KDR
- IDH1
- HTR1A
- HRH3
- HRH2
- NPY2R
- OPRD1
- HDAC6
- OPRK1
- TDP1
- TBXAS1
- TBXA2R
- TACR2
- TACR1
- SMAD3
- SLC6A4
- SLC6A3
- PTPRC
- PTGS2
- PTGS1
- PTAFR
- PRKCA
- PPP3CA
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ACM1
- ACM4
- ACM5
- ALR
- CP3A4
- GSTP1
- MCHR1
- MDM2
- MDM4
- NPBW1
- TNNC1
- TNNI3
- TNNT2
Cross-references
Synonyms
- pecazine
- mepazin
- mepazine base
- meprazine
- mesapin
- nothiazine
- mepazine acetate
- Pecazine
- Pecazina
- Lacumin
- Mepasin
- Mepazin
- Mepazine base
- Meprazine
- Mesapin
- Nothiazine
- Pacatal
- Pacatal base
- Pacatol
- Pakatal
- Paxital
- Pecatal
- III-2318
- P-391
- Pecazinum
- Pecazine [INN:BAN]
- Pecazinum [INN-Latin]
- Pecazina [INN-Spanish]
- (N-Methyl-3-piperidyl)methylphenothiazine
- EINECS 200-490-8
- UNII-PH34873A38
- AI3-50131
- MEPAZINE [MI]
- PECAZINE [INN]
- PECAZINE [WHO-DD]
- PH34873A38
- Phenothiazine, 10-((1-methyl-3-piperidyl)methyl)-
- DTXCID0026177
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