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METHSCOPOLAMINE
SynDRA canonical compound SYN0006651 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | CHRM3 |
|---|
| Mechanism of action | Acetylcholine receptor antagonist |
|---|
| Indication | peptic ulcer disease (PUD) |
|---|
| Disease area | gastroenterology |
|---|
All known targets
- CHRM3
- CHRM1
- CHRM2
- CHRM4
- CHRM5
- Chrm3
- HRH1
Mechanisms of action (all sources)
- Acetylcholine receptor antagonist
- CHRM1 ANTAGONIST
- CHRM3 ANTAGONIST
- CHRM2 ANTAGONIST
- CHRM3 MODULATOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ACHE
- ADORA3
- TBXA2R
- SLC6A4
- SLC6A3
- SLC6A2
- PTGS1
- PGR
- PDE4A
- PDE3A
- OPRM1
- MAOA
- KDR
- KCNH2
- HTR2B
- HTR1A
- HSD17B10
- HRH3
- HIF1A
- F2
- ESR1
- DRD3
- DRD1
- CYP3A4
- CYP2D6
- CYP2C9
- CYP2C19
- CYP1A2
- AR
- ADRA2A
- ADRA1A
- TSHR
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Cholinergic Antagonists
- Anticholinergic
- Parasympatholytics
- Peripheral Nervous System Agents
ATC classes
- A03B · BELLADONNA AND DERIVATIVES, PLAIN
- S01F · MYDRIATICS AND CYCLOPLEGICS
- ANTISPASMODICS IN COMBINATION WITH PSYCHOLEPTICS
Cross-references
Synonyms
- METHSCOPOLAMINE BROMIDE
- PAMINE
- PAMINE FORTE
- Pamine
- methylscopolamine
- N-Methylhyoscine
- N-Methylscopolamine
- methscopolamine bromide
- methscopolamine nitrate
- methylscopolamine bromide
- Methylscopolamine
- (-)-n-methylscopolamine
- Methscopolamine cation
- Methscopolamine ion
- N-methylhyoscine
- N-methylscopolamine
- Methscopolamine Bromide
- Pamine Forte
- N-methyl scopolamine
- UNII-VDR09VTQ8U
- VDR09VTQ8U
- CHEMBL376897
- Metylskopolamin
- HSDB 5420
- [3H]N-methylscopolamine
- [3H]N-methyl scopolamine
- [3H]NMS
- Methyl scopolamine
- 3C0
- CHEMBL3140030
- Methscopolamine (bromide)
- N-methylscopolamine (NMS)
- SCHEMBL65398
- GTPL316
- GTPL317
- METHSCOPOLAMINE [VANDF]
- DTXSID0046931
Reported adverse events
- Headache
- Nausea
- Tachycardia
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