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TIAPROFENIC ACID
SynDRA canonical compound SYN0005812 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | PTGS2 |
|---|
| Mechanism of action | Cyclooxygenase inhibitor |
|---|
| Indication | rheumatoid arthritis |
|---|
| Disease area | rheumatology |
|---|
All known targets
Mechanisms of action (all sources)
- Cyclooxygenase inhibitor
- PTGS2 INHIBITOR
- PTGS1 INHIBITOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- KCNH2
- DRD3
- NR1I2
- ADORA1
- HRH3
- HTR2A
- HTR2B
- HTR2C
- HTR3A
- MAOA
- MC3R
- MC4R
- MLNR
- NPY1R
- NR3C1
- OPRD1
- OPRK1
- OPRM1
- PDE3A
- PDE4D
- PGR
- SAMHD1
- SLC29A1
- SLC6A2
- SLC6A3
- SLC6A4
- TBXA2R
- TDP1
- UCHL5
- UGT2B10
- UGT2B4
- HTR1A
- HRH2
- ADORA2A
- HDAC6
- ADORA3
- ADRA1A
- ADRA2A
- ADRA2B
- ADRA2C
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- CASP1
- CASP3
- CASP4
- CASP5
- CASP9
- CP1A2
- CP2C9
- CP2CJ
- ESRRA
- HDAC9
- RARA
- SENP6
- SENP7
- SENP8
Drug classes
- Analgesics
- Analgesics, Non-Narcotic
- Anti-Inflammatory Agents
- Anti-Inflammatory Agents, Non-Steroidal
- Antirheumatic Agents
- Peripheral Nervous System Agents
- Sensory System Agents
ATC classes
- M01A · ANTIINFLAMMATORY AND ANTIRHEUMATIC PRODUCTS, NON-STEROIDS
Cross-references
Synonyms
- (RS)-Tiaprofenic acid
- (+/-)-Tiaprofenic acid
- tiaprofen
- Acide tiaprofenique
- Acido tiaprofenico
- Surgam
- Tiaprofen
- Tiaprofenate
- RU-15060
- Surgam 200
- Surgam 300
- Surgam sa
- Tiaprofensaeure
- Acidum tiaprofenicum
- Surgam SR
- FC 3001
- RU 15060
- Acide tiaprofenique [INN-French]
- Acido tiaprofenico [INN-Spanish]
- Acidum tiaprofenicum [INN-Latin]
- Apo-Tiaprofenic Tablets
- Dom-tiaprofenic
- Surgam (TN)
- Surgamyl (TN)
- Tiaprofen (TN)
- Tiaprofenic acid (JAN/INN)
- Tiaprofenic-200-Tab
- Tiaprofenic-300-Tab
- Tiaprofenic acid [INN:BAN:DCF:JAN]
- Alpha-methyl-5-benzoyl-2-thienylacetic acid
- 2-(5-Benzyl-2-thienyl)propionsaeure
- 2-(5-benzoylthiophen-2-yl)propanoic acid
- 2-[5-(phenylcarbonyl)-2-thienyl]propanoic acid
- 5-Benzoyl-alpha-methyl-2-thiopheneacetic acid
- 5-benzoyl-alpha-methylthiophene-2-acetic acid
- tiaprofenic-acid
- alpha-methyl-5-benzoyl-2-thienylacetic acid
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