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ARTESUNATE
SynDRA canonical compound SYN0005780 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx |
|---|
| Mechanism of action | DNA synthesis inhibitor |
|---|
| Indication | malaria |
|---|
| Disease area | infectious disease |
|---|
All known targets
- ATP1A1
- CYP2B6
- CYP2C19
- CYP3A5
Mechanisms of action (all sources)
- DNA synthesis inhibitor
- ATP1A1 BINDER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- PTGES2
- ADORA1
- NR3C1
- HTR1A
- HTR2A
- HTR2B
- HTR2C
- HTR3A
- KCNH2
- MAOA
- MC3R
- MLNR
- NPY1R
- NR1I2
- OPRD1
- ADORA2A
- OPRK1
- OPRM1
- PDE3A
- PDE4D
- PGR
- PTGS2
- SLC29A1
- SLC6A2
- SLC6A3
- SLC6A4
- TBXA2R
- HRH3
- HRH2
- HRH1
- CCKAR
- ADORA3
- ADRA1A
- ADRA2A
- ADRA2B
- ADRA2C
- ADRB1
- ADRB2
- AGTR1
- AVPR1A
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Anthelmintics
- Anti-Infective Agents
- Antimalarials
- Antineoplastic Agents
- Antiparasitic Agents
- Antiplatyhelmintic Agents
- Antiprotozoal Agents
- Antiviral Agents
- Schistosomicides
- Antimalarial
- antimalarial agent
ATC classes
Cross-references
Synonyms
- arinate
- arsuamoon
- arsumax
- artesunic acid
- cosunate
- dihydroqinghasu hemsuccinate
- artesunate amivas
- Artesunato
- .alpha.-artesunic acid
- Artesunatum
- Artesunic acid
- Dihydroqinghaosu hemisuccinate
- Plasmotrin
- Qinghaozhi
- Saphnate
- Zysunate
- LJPC-0118
- NSC-712571
- Arsumax
- Artesunate amivas
- Arinate
- Artsuna
- Dihydroqinghaosusuccinate
- Nuartez
- Plasmotrim
- Dihydroqinghasu hemsuccinate
- Quinghaosu reduced succinate ester
- Succinyl dihydroartemisinin
- SM 804
- WR-256283
- Arsumax (TN)
- Artesunate (USAN)
- Artesunate (superseded RN)
- Artesunato [INN-Spanish]
- Artesunatum [INN-Latin]
- Dihydroartemisinine-12-alpha-succinate
- Asumax
Reported adverse events
- Aspartate aminotransferase increased
- Chills
- Fatigue
- Hypersensitivity
- Infection
- Insomnia
- Malaise
- Nasopharyngitis
- Palpitations
- Plasmodium falciparum infection
- Pruritus
- Rhinitis
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