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GALLAMINE
SynDRA canonical compound SYN0005629 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · OTC |
|---|
| Primary target(s) | CHRM2 | CHRNA1 |
|---|
| Mechanism of action | acetylcholine receptor antagonist |
|---|
| Indication | muscle relaxant |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- CHRM2
- CHRNA1
- ACHE
- CHRM1
- CHRNB1
- CHRND
- CHRNG
- Chrm2
- ache
Mechanisms of action (all sources)
- CHRNA1 ANTAGONIST
- CHRNG ANTAGONIST
- CHRNB1 ANTAGONIST
- CHRND ANTAGONIST
- ACHE ANTAGONIST
- CHRM2 NEGATIVE ALLOSTERIC MODULATOR
- CHRNA1 MODULATOR
- acetylcholine receptor antagonist
- CHRM2 ANTAGONIST
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- KCNH2
- ADORA1
- LCK
- MMP9
- MMP1
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- MAPK1
- MAOA
- KDM4A
- FYN
- KAT2A
- HTR6
- HTR2C
- HTR2B
- HTR2A
- HRH2
- HRH1
- HMGCR
- MPHOSPH8
- NPY1R
- NPY2R
- NR3C1
- TBXAS1
- TACR2
- TACR1
- SLCO1B3
- SLCO1B1
- SLC6A4
- SLC6A3
- SLC6A2
- SIGMAR1
- PTPRC
- PTGS2
- PTGS1
- PTAFR
- PRKCA
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ACM2
- GNAI1
- NTM1A
- NTMT1
- RGS12
Drug classes
- Cholinergic Agents
- Cholinergic Antagonists
- Neuromuscular Agents
- Neuromuscular Blocking Agents
- Neuromuscular Nondepolarizing Agents
- Neurotransmitter Agents
- Nicotinic Antagonists
- Peripheral Nervous System Agents
ATC classes
- MUSCLE RELAXANTS, PERIPHERALLY ACTING AGENTS
Cross-references
Synonyms
- FLAXEDIL
- flaxedil
- gallamine triethochloride
- gallamonium iodide
- gallamine triethyl iodide
- gallamine triethiodide
- Gallamine Triethiodide
- Benzkurin
- Flaxedil
- Gallaflex
- Parexyl
- Pirolakson
- Pyrolaxon
- Relaxan
- Remyolan
- Retensin
- Sincurarine
- Syncurarine
- Tricuran
- Benzcurine iodide
- Gallamin triethiodide
- Gallamina triodoetilato
- Gallamina triodoetilato [DCIT]
- Gallamine iodide
- Gallamine triethiodide [INN]
- Gallamine triiodoethylate
- Gallamini triethiodidum
- Gallaminii iodidum
- Gallaminum triaethjodidum
- Gallaminum triaethoiodatum
- Gallamone triethiodide
- Gallamoni jodidum
- Miowas G
- Triethiodure de gallamine
- Triethiodurode galamina
- Triiodoethylate de gallamine
- Triiodoethylate de gallamine [French]
- F 2559
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