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DROPERIDOL
SynDRA canonical compound SYN0003759 — structure-anchored drug synonym record
| Clinical phase | Preclinical |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | DRD2 |
|---|
| Mechanism of action | Dopamine receptor antagonist |
|---|
All known targets
- DRD2
- DRD4
- DRD3
- HTR2A
- HTR1A
- SCN2A
- SCN1A
- Pgrmc1
- KCNH2
- Htr1a
- HTR4
- HTR2C
Mechanisms of action (all sources)
- Dopamine receptor antagonist
- HTR2A ANTAGONIST
- Serotonin 2a (5-HT2a) receptor antagonist
- DRD2 ANTAGONIST
- D2-like dopamine receptor antagonist
- DRD3 ANTAGONIST
- DRD4 ANTAGONIST
- DRD2 BINDER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ABCB11
- ESR1
- CACNA1C
- MAPT
- OPRD1
- NR3C1
- NPY2R
- NPY1R
- MMP9
- MMP1
- MC5R
- MC4R
- MC3R
- MAPK3
- OPRM1
- MAPK14
- MAPK1
- MAOA
- LMNA
- LCK
- KDR
- KDM4E
- HTR6
- HRH3
- HRH2
- OPRK1
- PDE3A
- HIF1A
- PDE4A
- TDP1
- TBXAS1
- TBXA2R
- TACR2
- TACR1
- SLCO1B3
- SLC6A4
- SLC6A3
- SLC6A2
- SIGMAR1
- SCN5A
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- CACNA1D
- CACNA1F
- CACNA1S
- CP2D6
- ESRRA
- KCMB1
- MDR1
- PPBT
- RXFP1
- UHRF1
Drug classes
- Adjuvants, Anesthesia
- Antiemetics
- Antipsychotic Agents
- Central Nervous System Agents
- Central Nervous System Depressants
- Dopamine Agents
- Dopamine Antagonists
- Dopamine D2 Receptor Antagonists
- Gastrointestinal Agents
- Neurotransmitter Agents
- Peripheral Nervous System Agents
- Psychotropic Drugs
ATC classes
Cross-references
Synonyms
- FENTANYL CITRATE AND DROPERIDOL
- INAPSINE
- INNOVAR
- dehydrobenzperidol
- droleptan
- inapsin
- inapsine
- neurolidol
- MCN-JR-4749
- NSC-169874
- R-4749
- Dridol
- Droleptan
- Droperidol component of innovar
- Inapsine
- DHBP
- Dehidrobenzperidol
- Dehydrobenzoperidol
- Dehydrobenzperidol
- Deidrobenzperidolo
- Dihidrobenzperidol
- Droperidolo
- Droperidolum
- Halkan
- Inappin
- Inapsin
- Innovan
- Inopsin
- Inoval
- Leptanal
- Leptofen
- Properidol
- Sintodril
- Sintosian
- Thalamanol
- Thalamonal
- Vetkalm
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