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ACETOPHENAZINE
SynDRA canonical compound SYN0003638 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · OTC |
|---|
| Primary target(s) | DRD1 | DRD2 |
|---|
| Mechanism of action | dopamine receptor antagonist |
|---|
| Indication | psychosis |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
Mechanisms of action (all sources)
- DRD2 ANTAGONIST
- Dopamine D2 receptor antagonist
- dopamine receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- HRH1
- ADRA2C
- HTR1A
- KCNH2
- DRD3
- HTR2B
- HTR2A
- ADRA2A
- ADRA1A
- ADRA2B
- NR3C1
- SLC6A4
- HTR2C
- HTR3A
- MAOA
- MC3R
- MLNR
- NR1I2
- SLC6A3
- SLC6A2
- OPRD1
- OPRM1
- PDE4D
- PGR
- PPARG
- PTGS2
- SLC29A1
- PDE3A
- ADORA1
- HRH3
- ADORA2A
- ADORA3
- ADRB1
- ADRB2
- AGTR1
- AVPR1A
- CCKAR
- CHRM1
- CHRM2
- CHRM3
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
ATC classes
Cross-references
Synonyms
- TINDAL
- acetofenazine
- acetofenazine maleate
- acetophenazine maleate
- tindal maleate
- tindal
- Acetofenazina
- Acephenazinum
- Acetophenazina
- Acetophenazinum
- Tindal
- Acetophenazine [INN]
- Acetophenazina [INN-Spanish]
- Acetophenazinum [INN-Latin]
- 2-acetyl-10-[3-[4-(b-hydroxyethyl)piperazinyl]propyl]phenothiazine
- CHEBI:2401
- Acetophenazine (dimaleate)
- 8620H6K4QH
- NCGC00181120-01
- UNII-8620H6K4QH
- ACETOPHENAZINE [MI]
- CHEMBL1085
- SCHEMBL94266
- ACETOPHENAZINE [VANDF]
- ACETOPHENAZINE [WHO-DD]
- DTXSID2022547
- BDBM82475
- NSC_17676
- ZINC22446634
- DB01063
- NCGC00181120-02
- CAS_5714-00-1
- HY-116916
- CS-0066801
- FT-0744314
- C06807
- 5-(HYDROXYMETHYL)-3-PYRIDINYLBORONICACID
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