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BEPRIDIL
SynDRA canonical compound SYN0003100 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · OTC |
|---|
| Primary target(s) | CACNA1C | KCNQ4 | SCN5A |
|---|
| Mechanism of action | calcium channel blocker |
|---|
| Indication | angina pectoris |
|---|
| Disease area | cardiology |
|---|
All known targets
- KCNQ4
- CACNA1C
- CACNA1A
- CACNA1D
- SCN5A
- CACNA1H
- CACNG6
- CACNG7
- CACNG8
- HCN4
- KCNH2
- SCN1A
Mechanisms of action (all sources)
- CACNA1H BLOCKER
- CACNA2D1 BLOCKER
- CACNA1C BLOCKER
- CACNA2D3 BLOCKER
- CACNA1S BLOCKER
- CACNA2D2 BLOCKER
- CACNA1D BLOCKER
- CACNA1A BLOCKER
- CACNA1B BLOCKER
- CACNA1G BLOCKER
- CACNA2D4 BLOCKER
- CACNA1I BLOCKER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- CYP2C19
- ADRB1
- ESR1
- NR1I2
- KCNK2
- NPY1R
- CYP2C9
- DRD3
- ADRB2
- ADRA2C
- ADRA2B
- OPRK1
- ADRA1A
- CNR1
- HRH1
- DRD2
- NPY2R
- NPSR1
- MLNR
- MC4R
- ABCB1
- MC3R
- MAPT
- MAOA
- KDM4E
- IDH1
- HTT
- HTR3A
- HTR2C
- HTR2B
- LMNA
- OPRD1
- NR3C1
- NTSR1
- TDP1
- TBXA2R
- SMPD1
- SMN1
- SLCO1B3
- SLCO1B1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- 5HT2A
- JUN
- SYK
- SC5A7
- RGS12
- RARA
- PRGR
- NTM1A
- NSD2
- NPBW1
- MDR1
- MDM4
- MDM2
- MCHR1
- M4K2
- KSYK
- IL1B
- ANDR
- IFNG
- IDHC
- HS90B
- HS90A
- GNAI1
- GLSK
- GLI3
- ESRRA
- CP3A7
- CP2D6
- CP2CJ
- CACNA1S
- CACNA1F
- APAF
- TP53
Drug classes
- Anti-Arrhythmia Agents
- Antihypertensive Agents
- Calcium Channel Blockers
- Calcium-Regulating Hormones and Agents
- Cardiovascular Agents
- Membrane Transport Modulators
- Vasodilator Agents
ATC classes
- C08E · NON-SELECTIVE CALCIUM CHANNEL BLOCKERS
Cross-references
Synonyms
- BEPADIN
- VASCOR
- bepridil hydrochloride hydrate
- bepridil hydrochloride
- dl-Bepridil
- (+/-)-Bepridil
- bepricol
- Org 5730
- bepridil monohydrochloride monohydrate
- bepridil monohydrochloride
- cordium
- bepridil HCl
- Bepadin
- Vascor
- CERM 1978
- Bepadin (TN)
- Bepridil (INN)
- Vascor (TN)
- CHEBI:3061
- DTXCID402663
- 1-(2-(N-BENZYLANILINO)-1-(ISOBUTOXYMETHYL)ETHYL)-PYRROLIDINE
- bepridilum
- Bedapin
- Bepridil, alpha
- RefChem:567017
- Monohydrochloride, Bepridil
- CERM1978
- Bepridil Monohydrochloride, alpha
- C08EA02
- Monohydrochloride, alpha-Isomer Bepridil
- N-Benzyl-N-(3-isobutoxy-2-(pyrrolidin-1-yl)propyl)aniline
- C24H34N2O
- NCGC00015155-03
- BEPRIDIL [INN]
- Org-5730
- Bepridil free base
- (+/-)-Bepridil;Org 5730; dl-Bepridil
- CAS-64706-54-3
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