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MEQUITAZINE
SynDRA canonical compound SYN0003094 — structure-anchored drug synonym record
| Primary target(s) | HRH1 |
|---|
| Mechanism of action | Histamine receptor antagonist |
|---|
All known targets
- HRH1
- CHRM1
- CHRM2
- CHRM3
- CHRM4
- CHRM5
- TPR
Mechanisms of action (all sources)
- Histamine receptor antagonist
- HRH1 ANTAGONIST
- Histamine H1 receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- HTR2A
- SLC6A2
- HTR3A
- HTR2B
- EGFR
- DRD1
- CHRNA4
- DRD2
- KCNH2
- ADRA1A
- ADRA2B
- ADRA2A
- OPRM1
- SNCA
- MAPT
- MC3R
- MLNR
- NPSR1
- NR1I2
- NR3C1
- OPRD1
- SLC6A3
- SLC29A1
- PDE4D
- PGR
- MAOA
- POLB
- SLC6A4
- POLI
- PPARG
- PTGS2
- PDE3A
- ADORA1
- KDR
- HTR2C
- ADORA3
- ADRA2C
- ADRB1
- ADRB2
- AGTR1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ACM1
- ACM4
- SYK
- SMAD3
- SMAD2
- RARA
- PRGR
- PPARD
- NPBW1
- MLLT3
- MDM4
- MDM2
- MCHR1
- KSYK
- KCNJ1
- GLI3
- GCR
- CP2D6
- CP19A
- CASP7
- CASP3
- BRCA1
- BARD1
- ATXN2
- ANDR
- ALR
- ACM5
- TERA
Drug classes
- Histamine Agents
- Histamine Antagonists
- Histamine H1 Antagonists
- Neurotransmitter Agents
ATC classes
- R06A · ANTIHISTAMINES FOR SYSTEMIC USE
Cross-references
Synonyms
- metaplexan
- nipolazin
- Mequitazina
- Kitazemin
- NSC-303612
- Primalan
- Butix
- Instotal
- Mequitazinum
- Metaplexan
- Mircol
- Quitadrill
- Vigigan
- Virginan
- Zesulan
- Italfarmaco brand of mequitazine
- Mequitazina [Spanish]
- Mequitazine hydrochloride
- Pierre Fabre brand of mequitazine
- LM-209
- Kitazemin (TN)
- Mequitazina [INN-Spanish]
- Mequitazinum [INN-Latin]
- Mequitazine (JP15/INN)
- Mequitazine [INN:BAN:DCF:JAN]
- Mequitazine tartrate, (R-(R*,R*))-isomer
- 10-(1-Azabicyclo[2.2.2]oct-3-ylmethyl)-10H-phenothiazine
- 10-(1-azabicyclo(2.2.2)oct-8-ylmethyl)phenothiazine
- 10-(1-azabicyclo[2.2.2]octan-3-ylmethyl)phenothiazine
- 10-(3-Quinuclidinylmethyl)phenothiazine
- 10H-Phenothiazine, 10-(1-azabicyclo(2.2.2)oct-3-ylmethyl)-(9CI)
- 3-Methylquinuclidinyl-10-phenothiazine
- levomequitazine
- NSC 303612
- Y463242LY2
- DTXCID303262
- RefChem:811005
- R06AD07
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