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PIPAMPERONE
SynDRA canonical compound SYN0002224 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | HTR2A |
|---|
| Mechanism of action | Dopamine receptor antagonist |
|---|
| Indication | schizophrenia |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- HTR2A
- DRD2
- HRH1
- HTR1A
- HTR1B
- HTR1D
- ADRA2A
- ADRA2B
- ADRA2C
- ADRB1
- ADRB2
- DRD3
Mechanisms of action (all sources)
- Dopamine receptor antagonist
- HTR1A ANTAGONIST
- HTR1B ANTAGONIST
- HTR1D ANTAGONIST
- HTR2A ANTAGONIST
- HRH1 ANTAGONIST
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ADRA1A
- SLC6A3
- DRD1
- KCNH2
- OPRM1
- ACHE
- PDE3A
- TBXA2R
- SLC6A4
- SLC6A2
- SLC47A2
- SLC47A1
- PTGS1
- PGR
- PDE4A
- MAOA
- ADORA3
- KDR
- HRH3
- F2
- ESR1
- CHRM2
- CHRM1
- AR
- APEX1
- TDP1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- 5HT1A
- 5HT1B
- 5HT1D
- 5HT2A
- CP2D6
Drug classes
- Antipsychotic Agents
- Central Nervous System Agents
- Central Nervous System Depressants
- Neurotransmitter Agents
- Psychotropic Drugs
- Serotonin Agents
- Serotonin Antagonists
- Tranquilizing Agents
ATC classes
Cross-references
Synonyms
- pipamperone dihydrochloride
- dipiperon
- dipiperone
- floropipamide
- dipiperal
- pipamperone hydrochloride
- pipamperone HCl
- Pipamperona
- Pipamperone hydrochloride
- Floropipamide
- Pipaneperone
- NSC-759178
- R-3345
- Dipiperon
- Dipiperone
- Dipiperal
- Piperonyl
- Piperonil
- Pipamperonum
- Pipamperone HCl
- McN-JR-3345
- R 3345
- Pipamperonum [INN-Latin]
- Pipamperona [INN-Spanish]
- Propitan
- Pipamperone [USAN:INN:BAN]
- CCRIS 9071
- UNII-5402501F0W
- BRN 0496532
- (1,4'-BIPIPERIDINE)-4'-CARBOXAMIDE, 1'-(3-(p-FLUOROBENZOYL)PROPYL)-
- CHEBI:78549
- p-Fluoro-gamma-(4-piperidino-4-carbamoylpiperidino)butyrophenone
- NSC 759178
- RefChem:863377
- DTXCID8028343
- N05AD05
- PIPAMPERONE DIHYDROCHLORIDE APPROX. 99
- Pipamperone free base
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