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TAMSULOSIN
SynDRA canonical compound SYN0002125 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | ADRA1A |
|---|
| Mechanism of action | Adrenergic receptor antagonist |
|---|
| Indication | benign prostatic hyperplasia (BPH) |
|---|
| Disease area | urology |
|---|
All known targets
- ADRA1A
- ADRA1B
- ADRA1D
- ADRA2A
- ADRA2C
- Adra1a
- Adra1d
- Adra2b
- DRD2
- DRD3
- HTR1A
- HTR7
Mechanisms of action (all sources)
- Adrenergic receptor antagonist
- ADRA1A ANTAGONIST
- Adrenergic receptor alpha-1 antagonist
- ADRA1D ANTAGONIST
- ADRA1B ANTAGONIST
- ADRA1A MODULATOR
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- OPRM1
- ADRB2
- KCNH2
- NR1I2
- HTR2B
- ADRB1
- SLC6A4
- SLC6A3
- HTR2C
- HTR3A
- TBXA2R
- MAOA
- MC3R
- MC4R
- MLNR
- NPY1R
- NR3C1
- OPRD1
- OPRK1
- HTR2A
- PDE3A
- PDE4D
- PGR
- PTGS2
- SLC29A1
- SLC6A2
- ADORA1
- HRH3
- ADORA2A
- HRH2
- ADORA3
- AGTR1
- AVPR1A
- AVPR2
- BDKRB2
- CCKAR
- CCKBR
- CHRM1
- CHRM2
- CHRM3
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- ANDR
- CP2D6
- CP3A4
- CP3A7
- GPR151
Drug classes
- Adrenergic alpha-Antagonists
- alpha-Adrenergic Blocker
- Adrenergic Agents
- Adrenergic alpha-1 Receptor Antagonists
- Adrenergic Antagonists
- Neurotransmitter Agents
- Urological Agents
ATC classes
- G04C · DRUGS USED IN BENIGN PROSTATIC HYPERTROPHY
Cross-references
Synonyms
- DUTASTERIDE AND TAMSULOSIN HYDROCHLORIDE
- FLOMAX
- Flomax
- JALYN
- Jalyn
- TAMSULOSIN HYDROCHLORIDE
- tamsulosin hydrochloride
- tamsulosin HCl
- LY-253352
- Tamsulosine
- Tamsulosina
- Tamsulon
- HGP-0412
- HIP-1402
- HIP1402
- Flowmax
- Harnal
- Tamsolusin
- Tamsulosinum
- Flomax (TN)
- Flomaxtra (TN)
- Tamsulon (TN)
- Tamsulosin (INN)
- Tamsulosin [INN:BAN]
- Tamsulosina [INN-Spanish]
- Tamsulosine [INN-French]
- Tamsulosinum [INN-Latin]
- Urimax (TN)
- G3P28OML5I
- (-)-Tamsulosin
- (r)-(-)-tamsulosin
- CHEBI:9398
- RefChem:56609
- DTXCID803631
- G04CA02
- Alna
- Josir
- Omnic
Reported adverse events
- Priapism
- Headache
- Syncope
- Dizziness
- Asthenia
- Nausea
- Rhinitis
- Stevens-Johnson syndrome
- Somnolence
- Cough
- Insomnia
- Pharyngitis
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