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BUTORPHANOL
SynDRA canonical compound SYN0001803 — structure-anchored drug synonym record
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | OPRM1 |
|---|
| Mechanism of action | Opioid receptor antagonist |
|---|
All known targets
Mechanisms of action (all sources)
- Opioid receptor agonist
- Opioid receptor antagonist
- OPRM1 PARTIAL AGONIST
- Mu opioid receptor partial agonist
- OPRK1 PARTIAL AGONIST
- Kappa opioid receptor partial agonist
- OPRD1 AGONIST
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ADORA1
- MC3R
- GHSR
- HRH1
- HRH2
- HRH3
- HTR1A
- HTR2A
- HTR2B
- HTR2C
- HTR3A
- KCNH2
- MAOA
- MLNR
- EDNRA
- NPY1R
- NR1I2
- NR3C1
- PDE3A
- PDE4D
- PGR
- PPARG
- PTGS2
- SLC29A1
- SLC6A2
- SLC6A3
- ESR1
- DRD3
- ADORA2A
- CCKAR
- ADORA3
- ADRA1A
- ADRA2A
- ADRA2B
- ADRA2C
- ADRB1
- ADRB2
- AGTR1
- AVPR1A
- AVPR2
Drug classes
- Analgesics
- Analgesics, Opioid
- Antitussive Agents
- Central Nervous System Agents
- Central Nervous System Depressants
- Narcotic Antagonists
- Narcotics
- Peripheral Nervous System Agents
- Respiratory System Agents
- Sensory System Agents
- Partial Opioid Agonists
- Competitive Opioid Antagonists
ATC classes
Cross-references
Synonyms
- BUTORPHANOL TARTRATE
- BUTORPHANOL TARTRATE PRESERVATIVE FREE
- STADOL
- STADOL PRESERVATIVE FREE
- Torbugesic
- Torphadine
- (-)-Butorphanol
- butorphanol tartrate
- BC-2627
- Butorfanol
- LEVO-BC-2627
- Beforal
- Butorphanolum
- Moradol
- Stadol
- Butorphanol tartrate
- Beforal (TN)
- Butorfanol [INN-Spanish]
- Butorphanolum [INN-Latin]
- L-BC 2627
- Moradol (TN)
- Butorphanol (USAN/INN)
- Butorphanol [USAN:BAN:INN]
- Levo-BC-2627
- (-)-17-(Cyclobutylmethyl)morphinan-3,14-diol
- (-)-N-cyclobutylmethyl-3,14-dihydroxymorphinan
- (-)-butorphanol
- 17-(CYCLOBUTYLMETHYL)MORPHINAN-3,14-DIOL
- butorphanol-(+)-tartrate
- levo-BC-2627
- QV897JC36D
- Morphinan-3,14-diol, 17-(cyclobutylmethyl)-
- CHEBI:3242
- butorfanolo
- BC 2627
- RefChem:56687
- DTXCID502714
- N02AF01
Reported adverse events
- NGS
- Abnormal dreams
- Anxiety
- Asthenia
- Epistaxis
- Hypertension
- Hypotension
- Rash
- Allodynia
- Adrenal insufficiency
- Androgen deficiency
- Death
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