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ESMOLOL
SynDRA canonical compound SYN0001764 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | ADRB1 |
|---|
| Mechanism of action | Adrenergic receptor antagonist |
|---|
| Indication | hypertension | ventricular tachycardia (VT) |
|---|
| Disease area | cardiology |
|---|
All known targets
Mechanisms of action (all sources)
- Adrenergic receptor antagonist
- ADRB1 ANTAGONIST
- Beta-1 adrenergic receptor antagonist
- ADRB2 ANTAGONIST
- Beta-2 adrenergic receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ACHE
- MAPK1
- NR1I2
- NPY2R
- NPY1R
- MMP9
- MMP1
- MLNR
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- MAOA
- HDAC6
- LCK
- KCNH2
- HTR6
- HTR3A
- HTR2C
- HTR2B
- HTR2A
- HTR1A
- HRH3
- HRH2
- HRH1
- NR3C1
- OPRD1
- OPRK1
- OPRM1
- TBXAS1
- TBXA2R
- TACR2
- TACR1
- SLC6A4
- SLC6A3
- SLC6A2
- SLC47A2
- SLC47A1
- SLC29A1
Drug classes
- Adrenergic beta-Antagonists
- beta-Adrenergic Blocker
- Adrenergic Agents
- Adrenergic Antagonists
- Adrenergic beta-1 Receptor Antagonists
- Neurotransmitter Agents
ATC classes
- C07A · BETA BLOCKING AGENTS
Cross-references
Synonyms
- BREVIBLOC
- BREVIBLOC DOUBLE STRENGTH IN PLASTIC CONTAINER
- BREVIBLOC IN PLASTIC CONTAINER
- Brevibloc
- ESMOLOL HYDROCHLORIDE
- ESMOLOL HYDROCHLORIDE DOUBLE STRENGTH IN PLASTIC CONTAINER
- ESMOLOL HYDROCHLORIDE IN PLASTIC CONTAINER
- brevibloc
- esmolol hydrochloride
- esmolol HCl
- ASL-8052-001
- ASL 8052-001
- Brevibloc (TN)
- Esmolol (INN)
- Esmolol [INN:BAN]
- Methyl p-[2-hydroxy-3-(isopropylamino)propoxy]hydrocinnamate
- Methyl p-(2-hydroxy-3-(isopropylamino)propoxy)hydrocinnamate
- (+-)-Esmolol
- (+-)-methyl p-(2-hydroxy-3-(isopropylamino)propoxy)hydrocinnamate
- MDY902UXSR
- methyl p-(2-hydroxy-3-(isopropylamino)propoxy)hydrocinnamate
- esmololum
- RefChem:56563
- CHEBI:4856
- DTXCID702995
- C07AB09
- (+/-)-esmolol
- MFCD00864566
- ESMOLOL [INN]
- NCGC00185766-01
- UNII-MDY902UXSR
- BRN 5287174
- SR-01000763706
- Esmolol Impurity 106
- ESMOLOL [VANDF]
- ESMOLOL [MI]
- ESMOLOL [WHO-DD]
- SCHEMBL3605
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