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BROMPERIDOL
SynDRA canonical compound SYN0001564 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | DRD2 |
|---|
| Mechanism of action | Dopamine receptor antagonist |
|---|
| Indication | schizophrenia |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- DRD2
- ADRA1A
- CHRM1
- CHRM2
- CHRM3
- CHRM4
- CHRM5
- DRD1
- DRD3
- DRD4
- HRH1
- SIGMAR1
Mechanisms of action (all sources)
- Dopamine receptor antagonist
- DRD2 ANTAGONIST
- Dopamine D2 receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- HTR1A
- ADRB2
- HTR2A
- KCNH2
- GHSR
- NR1I2
- OPRK1
- OPRM1
- ADRA2C
- SLC6A2
- SLC6A4
- SLC6A3
- HTR2B
- PDE4D
- PDE3A
- TBXA2R
- HTR3A
- IDH1
- PTGS2
- MAOA
- POLI
- MC3R
- MLNR
- NFE2L2
- NPY1R
- SAMHD1
- NR3C1
- OPRD1
- PGR
- HTR2C
- SLC29A1
- ADORA1
- ADORA2A
- CCKBR
- ADORA3
- ADRA2A
- ADRA2B
- ADRB1
- AGTR1
- ALOX15B
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- 5HT2A
- ACM1
- ANDR
- CP1A2
- CP2D6
- CP3A4
- ESRRA
- GLI3
- NSD2
- SC5A7
- SMAD2
- SMAD3
Drug classes
- Antipsychotic Agents
- Central Nervous System Agents
- Central Nervous System Depressants
- Psychotropic Drugs
- Tranquilizing Agents
ATC classes
Cross-references
Synonyms
- bromperidol hydrochloride
- bromperidol HCl
- tesoprel
- azurene
- bromoperidol
- impromen
- NSC-759275
- R 11,333
- R-11333
- Impromen
- Bromoperidol
- Tesoprel
- Azurene
- 4-(4-(4-bromophenyl)-4-hydroxypiperidin-1-yl)-1-(4-fluorophenyl)butan-1-one
- UNII-LYH6F7I22E
- Bromperidolum [INN-Latin]
- R 11333
- EINECS 233-943-3
- 4-(4-(4-Bromophenyl)-4-hydroxypiperidino)-4'-fluorobutyrophenone
- CC 2489
- BRN 1552256
- LYH6F7I22E
- 4-(4-(p-Bromophenyl)-4-hydroxypiperidino)-4'-fluorobutyrophenone
- RKLNONIVDFXQRX-UHFFFAOYSA-N
- 4-(4-(4-Bromophenyl)-4-hydroxy-1-piperidinyl)-1-(4-fluorophenyl)-1-butanone
- NCGC00016692-01
- CAS-10457-90-6
- Bromperidolum
- NSC 759275
- DTXCID102690
- bromperidolo
- RefChem:570410
- N05AD06
- C21H23BrFNO2
- SR-05000001811
- Bromperidol CRS
- Impromen (TN)
- Bromperidol [USAN:INN:BAN:JAN]
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