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BISOPROLOL
SynDRA canonical compound SYN0001293 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · Rx/OTC |
|---|
| Primary target(s) | ADRB1 |
|---|
| Mechanism of action | Adrenergic receptor antagonist |
|---|
| Indication | hypertension |
|---|
| Disease area | cardiology |
|---|
All known targets
Mechanisms of action (all sources)
- Adrenergic receptor antagonist
- ADRB1 ANTAGONIST
- Beta-1 adrenergic receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- ADORA1
- HTR3A
- NFKB1
- MLNR
- MC4R
- MC3R
- MAPK1
- MAOA
- LMNA
- KCNH2
- HTR2C
- ADORA2A
- HTR2B
- HTR2A
- HTR1A
- HRH3
- HRH2
- HRH1
- HDAC6
- GMNN
- NPY1R
- NPY2R
- NR3C1
- NTSR1
- TBXA2R
- TACR1
- SLC6A4
- SLC6A3
- SLC6A2
- SLC47A2
- SLC47A1
- SLC29A1
- SCN5A
- PTGS2
- POLK
- PGR
- PDE4D
- PDE3A
- OPRM1
- OPRK1
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Adrenergic beta-Antagonists
- beta-Adrenergic Blocker
- Adrenergic Agents
- Adrenergic Antagonists
- Adrenergic beta-1 Receptor Antagonists
- Antihypertensive Agents
- Cardiovascular Agents
- Neurotransmitter Agents
- Peripheral Nervous System Agents
- Sympatholytics
ATC classes
- C07A · BETA BLOCKING AGENTS
- BETA BLOCKING AGENTS AND THIAZIDES
- BETA BLOCKING AGENTS, OTHER COMBINATIONS
- ACE INHIBITORS, COMBINATIONS
Cross-references
Synonyms
- BISOPROLOL FUMARATE
- BISOPROLOL FUMARATE AND HYDROCHLOROTHIAZIDE
- ZEBETA
- ZIAC
- bisoprolol hemifumarate
- bisoprolol fumarate
- CL 297,939
- EMD-33-512
- Bisocor
- Bisoprololum
- Cardicor
- Concor
- Detensiel
- Emconcor
- Emcor
- Euradal
- Isoten
- Monocor
- Soloc
- Soprol
- Zebeta
- Bisoprolol fumerate
- Bisoprolol hemifumarate
- Bisoprololum [Latin]
- CL-297939
- Concor (TN)
- Concore (TN)
- EMD-33512
- Monocor (TN)
- Zebeta (TN)
- Bisoprolol (USAN/INN)
- Bisoprolol [USAN:BAN:INN]
- Y41JS2NL6U
- CHEBI:3127
- Bisoprololum (Latin)
- bisoprololo
- RefChem:5608
- Hydrochloride, Bisoprolol
Reported adverse events
- Bradycardia
- Rash
- Fatigue
- Asthma
- Dizziness
- Dry mouth
- Purpura
- Arthralgia
- Orthostatic hypotension
- Vertigo
- Erythema multiforme
- Stevens-Johnson syndrome
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