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PROCAINE
SynDRA canonical compound SYN0000882 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Approval status | Approved · OTC |
|---|
| Primary target(s) | HTR3A |
|---|
| Mechanism of action | HMGCR inhibitor |
|---|
| Indication | anesthetic |
|---|
| Disease area | neurology/psychiatry |
|---|
All known targets
- HTR3A
- SCN10A
- RYR1
- SCN9A
- SCN8A
- GRIN3A
- SCN7A
- SCN5A
- SCN4A
- SCN3A
- SCN2A
- SCN1A
Mechanisms of action (all sources)
- HMGCR INHIBITOR
- SCN1A BLOCKER
- Sodium channel alpha subunit blocker
- SCN5A BLOCKER
- SCN4A BLOCKER
- SCN7A BLOCKER
- SCN2A BLOCKER
- SCN9A BLOCKER
- SCN3A BLOCKER
- SCN11A BLOCKER
- SCN8A BLOCKER
- SCN10A BLOCKER
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- HRH3
- ACHE
- MAPK1
- NPY2R
- NPY1R
- NPSR1
- MMP9
- MMP1
- MLNR
- MC5R
- MC4R
- MC3R
- MAPK3
- MAPK14
- LCK
- NR3C1
- KCNH2
- KAT2A
- HTR6
- HTR2C
- HTR2B
- HTR2A
- HTR1A
- HRH2
- HRH1
- HDAC6
- GMNN
- NR1I2
- OPRD1
- FYN
- OPRK1
- TSHR
- TBXAS1
- TARDBP
- TACR2
- TACR1
- SLCO1B3
- SLCO1B1
- SLC6A4
- SLC6A2
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
Drug classes
- Anesthetics
- Anesthetics, Local
- Central Nervous System Agents
- Central Nervous System Depressants
- Peripheral Nervous System Agents
- Sensory System Agents
ATC classes
- N01B · ANESTHETICS, LOCAL
- S01H · LOCAL ANESTHETICS
- C05A · AGENTS FOR TREATMENT OF HEMORRHOIDS AND ANAL FISSURES FOR TOPICAL USE
Cross-references
Synonyms
- ACHROMYCIN
- NOVOCAIN
- PROCAINE HYDROCHLORIDE
- PROCAINE HYDROCHLORIDE W/ EPINEPHRINE
- RAVOCAINE AND NOVOCAIN W/ LEVOPHED
- RAVOCAINE AND NOVOCAIN W/ NEO-COBEFRIN
- TETRACYN
- diethylaminoethyl p-aminobenzoate
- procain
- spinocaine
- isocaine
- isocain
- herocaine
- irocaine
- procaine hydrochloride
- procaine HCl
- Procaina
- NSC-169497
- Solution of novocain
- Allocaine
- Anticort
- Anuject
- Duracaine
- Gerokit
- Gerovital
- Jenacain
- Jenacaine
- Nissocaine
- Norocaine
- Novocain
- Novocaine
- Procain
- Procainum
- Scurocaine
- Spinocaine
- Factor H3
- SP01
- SP01A
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