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OXATOMIDE
SynDRA canonical compound SYN0000668 — structure-anchored drug synonym record
| Clinical phase | Launched |
|---|
| Primary target(s) | HRH1 |
|---|
| Mechanism of action | Histamine receptor antagonist |
|---|
| Indication | allergic rhinitis |
|---|
| Disease area | allergy |
|---|
All known targets
- HRH1
- CHRM1
- DRD3
- HTR2A
- HTR2B
- P2RX7
Mechanisms of action (all sources)
- Histamine receptor antagonist
- HRH1 ANTAGONIST
- Histamine H1 receptor antagonist
Bioactivity evidence (ChEMBL activities table — not curator-asserted)
- KCNH2
- GHSR
- DRD1
- ADRA1A
- HTR2C
- DRD2
- ADRA2C
- CHRM3
- SLC6A4
- SLC6A3
- SLC6A2
- CHRM2
- OPRM1
- NR1I2
- NR2E1
- NR2C1
- NEIL1
- NPY1R
- NEIL2
- NR4A1
- MUTYH
- MPHOSPH8
- MLNR
- MC3R
- MBD4
- NR3C1
- ADORA1
- NR5A1
- NTHL1
- UNG
- TDP1
- TDG
- TBXA2R
- SMUG1
- RXRA
- PTGS2
- PMP22
- PKM
- PGR
- PDE4D
Screening evidence (raw PubChem HTS — uncurated, known false-positive rate)
- 5HT2A
- ESR2
- RXFP1
- RARA
- PRGR
- NSD2
- KSYK
- GLI3
- GCR
- ESRRA
- CP3A7
- ANDR
- CP3A4
- CP2D6
- CP2C9
- CP1A2
- CASP7
- CASP3
- CAC1H
- ATXN2
- SYK
Drug classes
- Anti-Allergic Agents
- Anti-Asthmatic Agents
- Histamine Agents
- Histamine Antagonists
- Histamine H1 Antagonists
- Neurotransmitter Agents
- Respiratory System Agents
ATC classes
- R06A · ANTIHISTAMINES FOR SYSTEMIC USE
Cross-references
Synonyms
- KW-4354
- R 35 443
- celtect
- celtomide
- Oxatomida
- Celtect
- Cobiona
- Dasten
- NSC-309710
- R 35,443
- R-35443
- Tinset
- Oxatimide
- Oxatomidum
- Oxetal
- CBMicro_024634
- O 9387
- R35443
- Celtect (TN)
- McN-JR 35443
- Oxatomida [INN-Spanish]
- Oxatomide (tinset)
- Oxatomidum [INN-Latin]
- Oxatomide (JAN/USAN/INN)
- Oxatomide [USAN:BAN:INN:JAN]
- 1-(3-(4-(Diphenylmethyl)-1-piperazinyl)propyl)-1,3-dihydro-2H-benzimidazol-2-one
- 1-(3-(4-(Diphenylmethyl)-1-piperazinyl)propyl)-2-benzimidazolinone
- 1-[3-(4-Benzhydryl-piperazin-1-yl)-propyl]-1,3-dihydro-benzoimidazol-2-one
- 1-[3-[4-(Diphenylmethyl)-1-piperazinyl]propyl]-1,3-dihydro-2H-benzimidazol-2-one
- 1-[3-[4-(Diphenylmethyl)-1-piperazinyl]propyl]-2-benzimidazolinone
- 3-[3-(4-benzhydrylpiperazin-1-yl)propyl]-1H-benzimidazol-2-one
- R 35443
- J31IL9Z2EE
- NSC 309710
- DTXCID2025181
- CHEBI:31943
- RefChem:857075
- R06AE06
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